BDBM383954 6-chloro-2-[[5-chloro-3- (trifluoromethyl)pyrazol-1- yl]methyl]-8- (trifluoromethyl)pyrido[1,2- a]pyrimidin-4-one::US10280165, Example 54

SMILES FC(F)(F)c1cc(Cl)n(Cc2cc(=O)n3c(Cl)cc(cc3n2)C(F)(F)F)n1

InChI Key InChIKey=CAZZSJVYBYNVAH-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383954   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Genentech

US Patent
LigandPNGBDBM383954(6-chloro-2-[[5-chloro-3- (trifluoromethyl)pyrazol-...)
Affinity DataEC50:  2.47E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
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