BDBM383938 2-[[5-chloro-3- (trifluoromethyl)pyrazol-1- yl]methyl]-6-[(1R,2R)-2- (hydroxymethyl)cyclopropyl]-7- methyl-pyrido[1,2-a]pyrimidin-4-one::US10280165, Example 36

SMILES Cc1ccc2nc(Cn3nc(cc3Cl)C(F)(F)F)cc(=O)n2c1[C@@H]1C[C@H]1CO

InChI Key InChIKey=ZIQAAZNDFSSJJV-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383938   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Genentech

US Patent
LigandPNGBDBM383938(2-[[5-chloro-3- (trifluoromethyl)pyrazol-1- yl]met...)
Affinity DataEC50:  126nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
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