BDBM383933 2-[[5-cyclopropyl-3- (trifluoromethyl)pyrazol-1- yl]methyl]-N-ethyl-4-oxo-pyrido[1,2- a]pyrimidine-6-carboxamide::US10280165, Example 20

SMILES CCNC(=O)c1cccc2nc(Cn3nc(cc3C3CC3)C(F)(F)F)cc(=O)n12

InChI Key InChIKey=DOOUMSLVIZLSHU-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383933   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Genentech

US Patent
LigandPNGBDBM383933(2-[[5-cyclopropyl-3- (trifluoromethyl)pyrazol-1- y...)
Affinity DataEC50:  7.40E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
Go to US Patent