BDBM383932 2-[[3-cyclopropyl-5- (trifluoromethyl)pyrazol-1- yl]methyl]-N-ethyl-7-methyl-4-oxo- pyrido[1,2-a]pyrimidine-6- carboxamide::US10280165, Example 18

SMILES CCNC(=O)c1c(C)ccc2nc(Cn3nc(cc3C(F)(F)F)C3CC3)cc(=O)n12

InChI Key InChIKey=HHUOPRJFKHUDCY-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383932   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Genentech

US Patent
LigandPNGBDBM383932(2-[[3-cyclopropyl-5- (trifluoromethyl)pyrazol-1- y...)
Affinity DataEC50:  1.62E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
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