BDBM382129 4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-biphenyl]-2-yl)methoxy) phenyl)butanoic Acid::US10273230, Compound of Example 7

SMILES OC(=O)CCCc1ccc(OCC2=C(CCCC2)c2ccc(cc2)C2CC2)cc1

InChI Key InChIKey=MQTLWULQQFNNGR-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 382129   

TargetFree fatty acid receptor 4(Human)
Piramal Enterprises

US Patent
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  275nMAssay Description:Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details
Go to US Patent

TargetFree fatty acid receptor 4(Human)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at FFA4 (unknown origin) expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed