BDBM382060 2-[5-[2-(cyclopropylmethoxy)-6- fluorophenyl]-1-methylimidazol- 4-yl]pyridine-4-carboxylic acid::US10273222, Example 122

SMILES Cn1cnc(c1-c1c(F)cccc1OCC1CC1)-c1cc(ccn1)C(O)=O

InChI Key InChIKey=ZBFLZYQTWARVNO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 382060   

TargetLysine-specific demethylase 2B(Human)
Celgene Quantscel Research

US Patent
LigandPNGBDBM382060(2-[5-[2-(cyclopropylmethoxy)-6- fluorophenyl]-1-me...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quantscel Research

US Patent
LigandPNGBDBM382060(2-[5-[2-(cyclopropylmethoxy)-6- fluorophenyl]-1-me...)
Affinity DataIC50: 5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2020
Entry Details
US Patent