BDBM372338 N-[(3-fluoro-4-methoxy- phenyl)methyl]-3,4-dimethyl- pyrimido[4',5':4,5]furo[2,3- c]pyridazin-8-amine::US10239887, Cpd. No. 75

SMILES COc1ccc(CNc2ncnc3c2oc2nnc(C)c(C)c32)cc1F

InChI Key InChIKey=DQZNRAHVIPBUFB-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372338   

TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM372338(US10239887, Cpd. No. 75 | N-[(3-fluoro-4-methoxy- ...)
Affinity DataEC50:  1.07E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
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