BDBM372320 2-[3-[[(7,9- dimethylpyrido[3',2':4,5]furo d[3,2-]pyrimidin-4- yl)amino]methyl]phenyl] propan-2-ol::US10239887, Cpd. No. 57

SMILES Cc1cc(C)c2c(n1)oc1c(NCc3cccc(c3)C(C)(C)O)ncnc21

InChI Key InChIKey=YFGQOYBNZXBYGD-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372320   

TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM372320(US10239887, Cpd. No. 57 | 2-[3-[[(7,9- dimethylpyr...)
Affinity DataEC50:  4.27E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
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