BDBM372304 4-(azetidin-1-yl)-8- chloro-7,9-dimethyl- pyrido[3',2':4,5]furo[3,2- d]pyrimidine hydrochloride::US10239887, Cpd. No. 42

SMILES Cc1nc2oc3c(ncnc3c2c(C)c1Cl)N1CCC1

InChI Key InChIKey=LZEGWRCOLVKPAS-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372304   

TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM372304(US10239887, Cpd. No. 42 | 4-(azetidin-1-yl)-8- chl...)
Affinity DataEC50:  269nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
Go to US Patent