BDBM371670 N-(6-fluoropyridin-2-yl)-4-(2-(thiazol-2-yl)-4-(trifluoromethyl)phenyl)chroman-7-sulfonamide::US10239869, Example 96

SMILES Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2nccs2)C(F)(F)F)n1

InChI Key InChIKey=WIJLUUOHOGAOEI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 371670   

TargetSodium channel protein type 9 subunit alpha(Human)
Lupin

US Patent

LigandBDBM371670(N-(6-fluoropyridin-2-yl)-4-(2-(thiazol-2-yl)-4-(tr...)Copy SMILESCopy InChI

Affinity DataIC50: 8nMAssay Description:HEK-293 cells overexpressing the channel of interest were seeded in a 96-well plate at a density of 30000 cells/well and incubated at 37° C./5% CO2 f...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/30/2019
Entry Details
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