BDBM371668 N-(pyrimidin-4-yl)-4-(2-(thiazol-2-yl)-4-(trifluoromethyl)phenyl)chroman-7-sulfonamide::US10239869, Example 94

SMILES FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)-c1nccs1

InChI Key InChIKey=OJCSIENXLFQIMD-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 371668   

TargetSodium channel protein type 9 subunit alpha(Human)
Lupin

US Patent

LigandBDBM371668(N-(pyrimidin-4-yl)-4-(2-(thiazol-2-yl)-4-(trifluor...)Copy SMILESCopy InChI

Affinity DataIC50: 3nMAssay Description:HEK-293 cells overexpressing the channel of interest were seeded in a 96-well plate at a density of 30000 cells/well and incubated at 37° C./5% CO2 f...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/30/2019
Entry Details
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