BDBM365239 1-{3-[6-(4-Methyl-pyridin- 2-ylamino)-2-phenyl- pyrimidin-4-yl]-piperidin- 1-yl}-ethanone::US9868720, No. 106

SMILES CC(=O)N1CCCC(C1)c1cc(Nc2cc(C)ccn2)nc(n1)-c1ccccc1

InChI Key InChIKey=WONRMGKFZOQRMC-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 365239   

TargetMitogen-activated protein kinase kinase kinase 12(Human)
Genentech

US Patent

LigandBDBM365239(US9868720, No. 106 | 1-{3-[6-(4-Methyl-pyridin- 2-...)Copy SMILESCopy InChI

Affinity DataKi:  30.7nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/10/2019
Entry Details
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