BDBM361401 (S)-3-((2- methylmorpholino) methyl)-N-(1H- pyrazolo[4,3-b]pyridin-3- yl)isothiazolo[4,5-b] pyridin-6-amine::US10221172, Example 59

SMILES C[C@H]1CN(Cc2nsc3cc(Nc4n[nH]c5cccnc45)cnc23)CCO1

InChI Key InChIKey=ZSLHEUZITPHWLA-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 361401   

TargetMetabotropic glutamate receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM361401((S)-3-((2- methylmorpholino) methyl)-N-(1H- pyrazo...)
Affinity DataEC50:  353nMAssay Description:In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...More data for this Ligand-Target Pair
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Date in BDB:
10/27/2019
Entry Details
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