BDBM361397 3-(morpholinomethyl)- N-(1H- pyrazolo[3,4-b]pyridin-3- yl)isothiazolo[4,5-b] pyridin-6-amine::US10221172, Example 55

SMILES C(N1CCOCC1)c1nsc2cc(Nc3n[nH]c4ncccc34)cnc12

InChI Key InChIKey=PXBAICMVSDYITR-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 361397   

TargetMetabotropic glutamate receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM361397(3-(morpholinomethyl)- N-(1H- pyrazolo[3,4-b]pyridi...)
Affinity DataEC50:  1.03E+3nMAssay Description:In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
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