BDBM358487 US10214544, Example 34

SMILES COC(=O)c1ccc(cc1)C(=O)Nc1cccc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(OC)sc3n2)c1

InChI Key InChIKey=ZUBMTRDIYXDCOO-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 358487   

TargetProteinase-activated receptor 4(Human)
Universite De Montreal

US Patent
LigandPNGBDBM358487(US10214544, Example 34)
Affinity DataEC50:  1.20nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent