BDBM355899 1-(4-(2- aminopyrimidin-4- yl)-3-chlorophenyl)- 3-(2-chloro-7- isopropylpyrazolo[1, 5-a]pyrimidin-6- yl)urea::US9815842, Example 23

SMILES CC(C)c1c(NC(=O)Nc2cnc(c(Cl)c2)-c2ccnc(N)n2)cnc2cc(Cl)nn12

InChI Key InChIKey=RJNVCKHFDBAILB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 355899   

TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Novartis

US Patent

LigandBDBM355899(US9815842, Example 23 | 1-(4-(2- aminopyrimidin-4-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
10/14/2019
Entry Details
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