BDBM355856 4-ethoxy-N-(3-fluoro-4-((5-(3-(2-hydroxypropan-2-yl)phenyl)pyrrolo[1,2-b]pyridazin-4-yl)oxy)phenyl)-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridin-3-carboxamide::US9815840, Example 43

SMILES CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnn3ccc(-c4cccc(c4)C(C)(C)O)c23)c(F)c1

InChI Key InChIKey=CXFRKQLSPSPVBM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 355856   

TargetHepatocyte growth factor receptor(Human)
The Asan Foundation

US Patent
LigandPNGBDBM355856(US9815840, Example 43 | 4-ethoxy-N-(3-fluoro-4-((5...)
Affinity DataIC50: 40nMAssay Description:The inhibitory effect of the compounds of the present invention on the activity of c-Met was confirmed as follows.Specifically, 250 μM G4Y1 pept...More data for this Ligand-Target Pair
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Date in BDB:
10/14/2019
Entry Details
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