BDBM350550 3-[(4- bromophenyl)carbamoyl] spiro[bicyclo[2.2.1]heptane- 7,1'-cyclopropane]-5-ene-2- carboxylic acid::US10208071, Compound 12::US10434112, Compound 12::US10799518, Compound 12

SMILES OC(=O)C1C2C=CC(C1C(=O)Nc1ccc(Br)cc1)C21CC1

InChI Key

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 350550   

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350550(3-[(4- bromophenyl)carbamoyl] spiro[bicyclo[2.2.1]...)
Affinity DataEC50:  4nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350550(3-[(4- bromophenyl)carbamoyl] spiro[bicyclo[2.2.1]...)
Affinity DataEC50:  4nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details
US Patent

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350550(3-[(4- bromophenyl)carbamoyl] spiro[bicyclo[2.2.1]...)
Affinity DataEC50:  4.00E+3nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
US Patent