BDBM350544 2-{[(2S)-2-{[(4- bromophenyl)carbamoyl] amino}-4- methylpentanoyl]amino}-2- methylpropanoic acid::US10208071, Compound 6::US10434112, Compound 6::US10799518, Compound 6

SMILES CC(C)C[C@H](NC(=O)Nc1ccc(Br)cc1)C(=O)NC(C)(C)C(O)=O

InChI Key InChIKey=WUZBUPYJADEKRK-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 350544   

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350544(2-{[(2S)-2-{[(4- bromophenyl)carbamoyl] amino}-4- ...)
Affinity DataEC50:  1.66E+3nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350544(2-{[(2S)-2-{[(4- bromophenyl)carbamoyl] amino}-4- ...)
Affinity DataEC50:  1.66E+3nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details
Go to US Patent

TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350544(2-{[(2S)-2-{[(4- bromophenyl)carbamoyl] amino}-4- ...)
Affinity DataEC50:  1nMAssay Description:Modulation of FPRL1 (unknown origin) expressed in CHO-Ga16 cells assessed as induction of calcium activity by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM350544(2-{[(2S)-2-{[(4- bromophenyl)carbamoyl] amino}-4- ...)
Affinity DataEC50:  1.66E+3nMAssay Description:HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent