BDBM350358 US9801878, 2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-ethyl]-6-methoxy-quinolinemethoxy-quinoline

SMILES COc1ccc2nc(CCc3nc4c(OC)ccc(C)n4n3)ccc2c1

InChI Key InChIKey=SFRANCVRDNUNDW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 350358   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
H. Lundbeck

US Patent

LigandBDBM350358(US9801878, 2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-...)Copy SMILESCopy InChI

Affinity DataIC50: 12nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
10/1/2019
Entry Details
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