BDBM350001 (R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benzo[d]imidazol-2-yl)methyl)-3- (3-(trifluoromethyl)phenyl) propanamide::US10208023, No. 75

SMILES N[C@H](Cc1cccc(c1)C(F)(F)F)C(=O)NCc1nc2c(cc(cc2[nH]1)C(F)(F)F)C(F)(F)F

InChI Key InChIKey=UPQWOERKVOUYPS-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 350001   

LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent