BDBM345480 N-[2-(2,4-Dichloro-6-methyl- phenoxy)-6-(1,5-dimethyl-6-oxo- 1,6-dihydro-pyridin-3-yl)-pyrimidin- 4-yl]-methanesulfonamide::US10202360, Example 25

SMILES Cc1cc(Cl)cc(Cl)c1Oc1nc(NS(C)(=O)=O)cc(n1)-c1cc(C)c(=O)n(C)c1

InChI Key InChIKey=FJOLCPBQPKTSHQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 345480   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM345480(US10202360, Example 25 | N-[2-(2,4-Dichloro-6-meth...)
Affinity DataIC50: 500nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
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