BDBM328406 6-chloro-3-(difluoromethyl)-1-((4-methoxy-3-(piperazin-1-yl) phenyl)sulfonyl)-1H-indazole::US9663498, Example 56

SMILES COc1ccc(cc1N1CCNCC1)S(=O)(=O)n1nc(C(F)F)c2ccc(Cl)cc12

InChI Key InChIKey=DCTJGGAVYMUWLI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 328406   

Target5-hydroxytryptamine receptor 6(Human)
Sunshine Lake Pharma

US Patent
LigandPNGBDBM328406(US9663498, Example 56 | 6-chloro-3-(difluoromethyl...)
Affinity DataIC50: 1.10nMAssay Description:The binding affinity of the compound of this invention to human 5-HT6 receptor expressed in CHO cell was evaluated by radioligand binding assay as fo...More data for this Ligand-Target Pair
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Date in BDB:
6/4/2019
Entry Details
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