BDBM328398 6-chloro-1-((3-(4-cyclobutylpiperazin-1-yl)-4-methoxyphenyl) sulfonyl)-3-(difluoromethyl)-1H-indole::US9663498, Example 41

SMILES COc1ccc(cc1N1CCN(CC1)C1CCC1)S(=O)(=O)n1cc(C(F)F)c2ccc(Cl)cc12

InChI Key InChIKey=OLSKECRQQAUTFF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 328398   

Target5-hydroxytryptamine receptor 6(Human)
Sunshine Lake Pharma

US Patent
LigandPNGBDBM328398(US9663498, Example 41 | 6-chloro-1-((3-(4-cyclobut...)
Affinity DataIC50: 0.5nMAssay Description:The binding affinity of the compound of this invention to human 5-HT6 receptor expressed in CHO cell was evaluated by radioligand binding assay as fo...More data for this Ligand-Target Pair
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Date in BDB:
6/4/2019
Entry Details
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