BDBM324017 US10189816, Compound 10

SMILES Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)C(O)=O)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O

InChI Key InChIKey=XGEUSSWNPIZVAK-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 324017   

TargetEnvelope glycoprotein gp160(HIV-1)
Viiv Healthcare UK (NO.5)

US Patent
LigandPNGBDBM324017(US10189816, Compound 10)
Affinity DataEC50: >1.00E+3nMAssay Description:A recombinant NL-RLuc proviral clone was constructed in which a section of the nef gene from NL4-3 was replaced with the Renilla Luciferase gene. Thi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

TargetEnvelope glycoprotein gp160(HIV-1)
Viiv Healthcare UK (NO.5)

US Patent
LigandPNGBDBM324017(US10189816, Compound 10)
Affinity DataEC50:  1.48E+3nMAssay Description:A recombinant NL-RLuc proviral clone was constructed in which a section of the nef gene from NL4-3 was replaced with the Renilla Luciferase gene. Thi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent