BDBM321451 3-[6-(cyclopropylmethyl)-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl]-N,N-dimethyl-benzamide::US10183009, Example 17

SMILES CN(C)C(=O)c1cccc(c1)-c1cn(CC2CC2)c(=O)c2[nH]ccc12

InChI Key InChIKey=FKGHEWSQSQHUQH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 321451   

TargetChromatin remodeling regulator CECR2 [424-538](Human)
Genentech

US Patent
LigandPNGBDBM321451(3-[6-(cyclopropylmethyl)-7-oxo-1H-pyrrolo[2,3-c]py...)
Affinity DataIC50: 5.60E+3nMAssay Description:His/Flag epitope tagged TAF1-BD21504-1635 was cloned, expressed, and purified to homogeneity. TAF1-BD2 binding and inhibition was assessed by monitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
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