BDBM321440 Ac-Arg-cyclo(Asp-Dab- D-Phe-Arg-Trp-Lys)- NH-cyclopropyl::US10179804, Example 122

SMILES CC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H]1CC(=O)CCCCC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CCN)NC1=O)C(=O)NC1CC1

InChI Key InChIKey=RMZNFIGKXAXQBU-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 321440   

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM321440(US10179804, Example 122 | Ac-Arg-cyclo(Asp-Dab- D-...)
Affinity DataKi:  3nMAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
Go to US Patent