BDBM310260 US10150760, Example 56.0::US10150760, Example 57.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc([C@H]2CCOC2)n1-c1c(OC)cccc1OC)c1ncc(Cl)cn1

InChI Key InChIKey=ZESIGRKAUDKULB-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 310260   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310260(US10150760, Example 56.0 | US10150760, Example 57....)
Affinity DataEC50:  19nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310260(US10150760, Example 56.0 | US10150760, Example 57....)
Affinity DataEC50:  21nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent