BDBM309994 US9657003, Bicalutamide

SMILES CC(O)(CS(=O)(=O)c1ccc(F)cc1)C(=O)CNc1ccc(C#N)c(c1)C(F)(F)F

InChI Key InChIKey=QOJLVADWVZTUIH-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 309994   

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309994(US9657003, Bicalutamide)
Affinity DataIC50: 228nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309994(US9657003, Bicalutamide)
Affinity DataKi:  40nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent