BDBM309987 N-((S)-1-(3-(3-chloro-4-cyano-2-methylphenyl)-1H-pyrazol-1-yl)propan-2-yl)-2-(1-hydroxyethyl)thiazole-4-carboxamide::US9657003, 186

SMILES C[C@@H](Cn1ccc(n1)-c1ccc(C#N)c(Cl)c1C)NC(=O)c1csc(n1)C(C)O

InChI Key InChIKey=ICFVJJDWCCMHPP-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 309987   

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309987(US9657003, 186 | N-((S)-1-(3-(3-chloro-4-cyano-2-m...)
Affinity DataIC50: 11nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309987(US9657003, 186 | N-((S)-1-(3-(3-chloro-4-cyano-2-m...)
Affinity DataKi:  3nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent