BDBM300977 6-((6S,8R)-7- (2,2- difluoroethyl)- 8-methyl- 6,7,8,9- tetrahydro-3H- pyrazolo[4,3- f]isoquinolin- 6-yl)-N-(1-(3- fluoropropyl) azetidin-3-yl)- N- methylpyridin- 3-amine::US10131663, Example 43::US10590130, Example 43::US10961241, Example 43

SMILES C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@H](N1CC(F)F)c1ccc(cn1)N(C)C1CN(CCCF)C1

InChI Key InChIKey=KETIMUXEJZGZHT-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 300977   

TargetEstrogen receptor(Human)
Astrazeneca

US Patent
LigandPNGBDBM300977(6-((6S,8R)-7- (2,2- difluoroethyl)- 8-methyl- 6,7,...)
Affinity DataIC50: 4.10nMAssay Description:The assay principle is that ER alpha-LBD (GST) is added to a fluorescent ligand to form a receptor/fluorophore complex. A terbium-labelled anti-GST a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetEstrogen receptor(Human)
Astrazeneca

US Patent
LigandPNGBDBM300977(6-((6S,8R)-7- (2,2- difluoroethyl)- 8-methyl- 6,7,...)
Affinity DataIC50: 0.25nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

LigandPNGBDBM300977(6-((6S,8R)-7- (2,2- difluoroethyl)- 8-methyl- 6,7,...)
Affinity DataIC50: 4.10nMAssay Description:hERG (human ether go go-related gene) potassium channels are essential for normal electrical activity in the heart. Arrhythmia can be induced by a bl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2020
Entry Details
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TargetEstrogen receptor [307-554](Human)
Astrazeneca

US Patent
LigandPNGBDBM300977(6-((6S,8R)-7- (2,2- difluoroethyl)- 8-methyl- 6,7,...)
Affinity DataIC50: 4.10nMAssay Description:The assay was performed as follows with all reagent additions carried out using the Beckman Coulter BioRAPTR FRD microfluidic workstation:1. Acoustic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2021
Entry Details
Go to US Patent