BDBM30057 triazolothiadiazine, 5I

SMILES COc1ccc(cc1OC)C1=Nn2c(SC1)nnc2-c1ccccc1C

InChI Key InChIKey=SZSOQWWQFQARJA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 30057   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Nih

LigandBDBM30057(triazolothiadiazine, 5I)Copy SMILESCopy InChI

Affinity DataIC50: 141nMpH: 7.2 T: 2°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In Depth
Date in BDB:
7/4/2009
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