BDBM299618 6-(3-isoprapoxy- phenyl) pyrido[3,2-d] pyrimidin-4- amine::US9592235, Example 365::US9855269, Compound 345

SMILES CC(C)Oc1cccc(c1)-c1ccc2ncnc(N)c2n1

InChI Key InChIKey=PVZAXFUSCQYMJR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 299618   

LigandPNGBDBM299618(US9592235, Example 365 | 6-(3-isoprapoxy- phenyl) ...)
Affinity DataIC50: 179nMAssay Description:The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
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LigandPNGBDBM299618(US9592235, Example 365 | 6-(3-isoprapoxy- phenyl) ...)
Affinity DataIC50: 179nMAssay Description:The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
Go to US Patent