BDBM296166 2-[4-[N-methyl-3-[methyl-(1- methylpiperidin-4- yl)amino]anilino]phenoxy]pyrido[3,4- d]pyrimidin-4-ol::US10112940, Example 89::US10202381, Example 89::US10208039, Example 89::US10611763, Example 89::US10815234, Example 89::US11535616, Example 89

SMILES CN(C1CCN(C)CC1)c1cccc(c1)N(C)c1ccc(Oc2nc(O)c3ccncc3n2)cc1

InChI Key InChIKey=DCEPDRIEVVJKJY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296166   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296166(US10112940, Example 89 | 2-[4-[N-methyl-3-[methyl-...)
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296166(US10112940, Example 89 | 2-[4-[N-methyl-3-[methyl-...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
Go to US Patent