BDBM296147 2-[4-[4-(4-aminobutan-2-yl)-N- methylanilino]phenoxy]pyrido[3,4- d]pyrimidin-4-ol::US10112940, Example 71::US10202381, Example 71::US10208039, Example 71::US10611763, Example 71::US10815234, Example 71::US11535616, Example 71

SMILES CC(CCN)c1ccc(cc1)N(C)c1ccc(Oc2nc(O)c3ccncc3n2)cc1

InChI Key InChIKey=GNLRAKTZEOBREI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296147   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296147(US10112940, Example 71 | 2-[4-[4-(4-aminobutan-2-y...)
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
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TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296147(US10112940, Example 71 | 2-[4-[4-(4-aminobutan-2-y...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
Go to US Patent