BDBM296101 2-{4-[methyl-(1,2,3,4-tetrahydro- naphthalen-1-ylmethyl)-amino]-phenoxy}- pyrido[3,4-d]pyrimidin-4-ol::US10112940, Example 28::US10202381, Example 28::US10208039, Example 28::US10611763, Example 28::US10815234, Example 28::US11535616, Example 28

SMILES CN(CC1CCCc2ccccc12)c1ccc(Oc2nc(O)c3ccncc3n2)cc1

InChI Key InChIKey=VJRRSIKXEUZPHL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296101   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296101(US10112940, Example 28 | 2-{4-[methyl-(1,2,3,4-tet...)
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296101(US10112940, Example 28 | 2-{4-[methyl-(1,2,3,4-tet...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
Go to US Patent