BDBM294252 Cis-N-(1-(3-(azetidin-1-yl)-4-benzyl-7-fluorochroman-6-yl)azetidin-3-yl)pyridazine-3-sulfonamide::US9586945, 9

SMILES Fc1cc2OCC(C(Cc3ccccc3)c2cc1N1CC(C1)NS(=O)(=O)c1cccnn1)N1CCC1

InChI Key InChIKey=QGPFUUSJRANRFB-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 294252   

TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Human)
Abbvie Deutschland

US Patent

LigandBDBM294252(US9586945, 9 | Cis-N-(1-(3-(azetidin-1-yl)-4-benzy...)Copy SMILESCopy InChI

Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/2/2019
Entry Details
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