BDBM293968 US10106552, Compound 43

SMILES NC(=O)c1sc2nc3C4CCC(C4)c3c(-c3cncs3)c2c1N

InChI Key InChIKey=GCTVOQIIGJKEBA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293968   

TargetEukaryotic elongation factor 2 kinase(Human)
Longevica Pharmaceuticals

US Patent
LigandPNGBDBM293968(US10106552, Compound 43)
Affinity DataIC50: 900nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
Go to US Patent