BDBM293926 US10106552, Compound 1

SMILES CC1(C)C\C(=C/c2ccc(Cl)o2)c2nc3sc(C(N)=O)c(N)c3c(-c3ccc(Cl)o3)c2C1

InChI Key InChIKey=GGLZTVNRCJRNMR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293926   

TargetEukaryotic elongation factor 2 kinase(Human)
Longevica Pharmaceuticals

US Patent
LigandPNGBDBM293926(US10106552, Compound 1)
Affinity DataIC50: 2.70E+3nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
Go to US Patent