BDBM293304 US10106504, Example 41

SMILES Cc1ccc(cc1)-c1c([C@H](OC(C)(C)C)C(O)=O)c(C)nc(C)c1-c1ccc2CN(Cc3c(C)cccc3F)CCc2c1

InChI Key InChIKey=LUTZYLHZBIURKZ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293304   

TargetGag-Pol polyprotein [489-587,Q496K](Human immunodeficiency virus type 1)
Viiv Healthcare UK (NO.5)

US Patent
LigandPNGBDBM293304(US10106504, Example 41)
Affinity DataEC50: <100nMpH: 7.55Assay Description:A recombinant NL-RLuc proviral clone was constructed in which a section of the nef gene from NL4-3 was replaced with the Renilla Luciferase gene. Thi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
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