BDBM28973 2-{1-[(4-chlorobenzene)sulfonyl]-4-[(trifluoromethane)sulfonylmethyl]cyclohexyl}-1,4-difluorobenzene::cyclohexyl sulfone-based compound, 17
SMILES Fc1ccc(F)c(c1)[C@]1(CC[C@H](CS(=O)(=O)C(F)(F)F)CC1)S(=O)(=O)c1ccc(Cl)cc1
InChI Key InChIKey=BCIWPZDEVCOVHV-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 28973
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Human)
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 21.5nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
