BDBM28926 (2S)-N-(5-chlorothiophen-2-yl)-5,5,5-trifluoro-1-hydroxy-3-(2,2,2-trifluoroethyl)pentane-2-sulfonamido::Begacestat analogue, 10
SMILES OC[C@@H](NS(=O)(=O)c1ccc(Cl)s1)C(CC(F)(F)F)CC(F)(F)F
InChI Key InChIKey=CJEZEJKUSJGLHH-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 28926
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Human)
Wyeth Research
Wyeth Research
Affinity DataEC50: 16nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair