BDBM289100 (−)-6-{4-[(3-Chloro-5-methylpyridin-2-yl)oxy]-2-methylphenyl}-1,5-dimethylpyrimidine-2,4(1H,3H)-dione (10)::US10093655, Example 10

SMILES Cc1cnc(Oc2ccc(c(C)c2)-c2c(C)c(=O)[nH]c(=O)n2C)c(Cl)c1

InChI Key InChIKey=QDDZCKNTJUFORZ-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289100   

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandPNGBDBM289100(US10093655, Example 10 | (−)-6-{4-[(3-Chloro...)
Affinity DataKi:  82.3nMpH: 7.4Assay Description:The affinity of the compounds described herein was determined by competition binding assays similar to those described in Ryman-Rasmussen et al., "Di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
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