BDBM285585 3-(4-chlorophenyl)-N-(5-methyl-1,2-oxazol-3-yl)imidazo[1,2-b]pyridazine-2-carboxamide,trifluoroacetate salt::US10077269, Example 58::US10669279, Example 58::US9598421, Example 58

SMILES Cc1cc(NC(=O)c2nc3cccnn3c2-c2ccc(Cl)cc2)no1

InChI Key InChIKey=WFHCBSIMFWEHOP-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 285585   

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 43.3nMAssay Description:Human PDE4A3 coding sequence (amino acids 2 to 825 from the sequence with accession number NP_001104779) was cloned into the baculovirus expression v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
US Patent

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 43.3nMAssay Description:The PDE4A3, PDE4B1, PDE4C1 and PDE4D3 assays use the Scintillation Proximity Assay (SPA) technology to measure the inhibition of human recombinant PD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details
US Patent

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 43.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 831nMAssay Description:Human PDE4A3 coding sequence (amino acids 2 to 825 from the sequence with accession number NP_001104779) was cloned into the baculovirus expression v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
US Patent

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 831nMAssay Description:The PDE4A3, PDE4B1, PDE4C1 and PDE4D3 assays use the Scintillation Proximity Assay (SPA) technology to measure the inhibition of human recombinant PD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details
US Patent

LigandPNGBDBM285585(US10077269, Example 58 | 3-(4-chlorophenyl)-N-(5-m...)
Affinity DataIC50: 831nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent