BDBM272996 (S)-2-(4-(1-(2- aminooxazolo[4,5- b]pyridin-5-yl)- 7,8,9,10-tetrahydro-6- oxa-2,10a- diazacycloocta[cd]inden- 4-yl)-1H-pyrazol-1- yl)butanamide::US10065970, Example 301::US10065970, Example 311::US10435414, Example 301

SMILES CC[C@@H](C(N)=O)n1cc(cn1)-c1cc2OCCCCn3c(nc(c1)c23)-c1ccc2oc(N)nc2n1

InChI Key InChIKey=ZLEHWGCPYUIMLF-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 272996   

LigandPNGBDBM272996((S)-2-(4-(1-(2- aminooxazolo[4,5- b]pyridin-5-yl)-...)
Affinity DataKi:  0.0310nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
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LigandPNGBDBM272996((S)-2-(4-(1-(2- aminooxazolo[4,5- b]pyridin-5-yl)-...)
Affinity DataKi:  0.0380nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
Go to US Patent

LigandPNGBDBM272996((S)-2-(4-(1-(2- aminooxazolo[4,5- b]pyridin-5-yl)-...)
Affinity DataKi:  0.0380nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
Go to US Patent