BDBM272909 (S)-2-((1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10- tetrahydro-6-oxa- 2,10a- diazacycloocta[cd]- inden-4-yl)amino)-2- cyclopropylacetamide::US10065970, Compound 214

SMILES NC(=O)[C@@H](Nc1cc2OCCCCn3c(nc(c1)c23)-c1ccc2nc(N)sc2c1)C1CC1

InChI Key InChIKey=FPXHUCUQLKQDIE-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 272909   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Genentech

US Patent

LigandBDBM272909((S)-2-((1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10...)Copy SMILESCopy InChI

Affinity DataKi: <0.0200nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/11/2018
Entry Details
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