BDBM27167 1H-indol-1-yl tertiary amine, 11::{[2-chloro-3-(trifluoromethyl)phenyl]methyl}[3-({4,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}oxy)propyl](2,2-diphenylethyl)amine

SMILES Cc1cc(C)c2c(OCCCN(CC(c3ccccc3)c3ccccc3)Cc3cccc(c3Cl)C(F)(F)F)n[nH]c2n1

InChI Key InChIKey=UIUZIKMYVPKHET-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 27167   

LigandPNGBDBM27167({[2-chloro-3-(trifluoromethyl)phenyl]methyl}[3-({4...)
Affinity DataEC50: >3.00E+3nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed
LigandPNGBDBM27167({[2-chloro-3-(trifluoromethyl)phenyl]methyl}[3-({4...)
Affinity DataEC50:  510nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2009
Entry Details Article
PubMed