BDBM271461 2-(6-((1H-indol-1-yl)sulfonyl)-4-hydroxy-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamido)acetic acid::US10065928, Example 7

SMILES Cn1c2ccc(cc2c(O)c(C(=O)NCC(O)=O)c1=O)S(=O)(=O)n1ccc2ccccc12

InChI Key InChIKey=ATLWTOYGAYAIMR-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 271461   

TargetHypoxia-inducible factor 1-alpha(Human)
Sunshine Lake Pharma

US Patent
LigandPNGBDBM271461(2-(6-((1H-indol-1-yl)sulfonyl)-4-hydroxy-1-methyl-...)
Affinity DataEC50:  6.83E+3nMAssay Description:The activities of compounds of the invention in inducing erythropoietin (EPO) production were assessed by using human live cancer cell strain Hep3B (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent