BDBM26724 N-[4-(quinolin-2-yl)phenyl]-1-(thiophene-2-sulfonyl)piperidine-4-carboxamide::quinoline analogue, 16e

SMILES O=C(Nc1ccc(cc1)-c1ccc2ccccc2n1)C1CCN(CC1)S(=O)(=O)c1cccs1

InChI Key InChIKey=RZVHGFPXYYBMTM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 26724   

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Abbott Laboratories

LigandPNGBDBM26724(N-[4-(quinolin-2-yl)phenyl]-1-(thiophene-2-sulfony...)
Affinity DataIC50: 21nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed