BDBM255719 US9475815, 104

SMILES COc1cc(C)cc2cc(sc12)-c1cc(C(=O)N2CCC[C@@H](N)C2)n2ncnc(N)c12

InChI Key InChIKey=FWTXUOUEFWFGHY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 255719   

TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Human)
Bayer Intelletual Property

US Patent
LigandPNGBDBM255719(US9475815, 104)
Affinity DataIC50: 14.6nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1 [400-80]/Glutathione S-transferase P(Human)
Bayer Intelletual Property

US Patent
LigandPNGBDBM255719(US9475815, 104)
Affinity DataIC50: 28.1nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-1 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2017
Entry Details
Go to US Patent